Pyrroloimidazolediones Derived from Aminomalonates and Benzaldehydes
نویسندگان
چکیده
Abstract Bicyclic lactams can be prepared from diethyl aminomalonate and substituted benzaldehydes by formation of a dimerised imidazolidine cycloadduct followed Dieckmann ring closure. The resulting N,N-heterocycles are metal-chelating but show no antibacterial activity.
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ژورنال
عنوان ژورنال: Synlett
سال: 2021
ISSN: ['0936-5214', '1437-2096']
DOI: https://doi.org/10.1055/s-0040-1720888